G-protein-coupled receptors (GPCRs) show great potential as molecular targets for the development of new therapeutics. These receptors play crucial roles in regulating numerous physiological processes such as learning and memory, immunity, cell actions, and development. Currently, licensed medications are only targeting certain types of GPCRs, while there are still many other GPCRs that have not been fully characterized. For this reason, a comprehensive investigation of GPCRs is urgent for drug development.
Fig.1 The signaling pathways of Gα protein-coupled GPCR.1
Creative Biolabs provides cost-effective Magic™ in vitro cell-based GPCR functional assay services that encompass multiple second messenger pathways for global customers to aid in drug development.
Our Magic™ in vitro cell-based GPCR functional assay services are characterized as the various second messengers' readouts according to the natural pathways of GPCRs. Our assays allow for the analysis of the candidate compounds and their regulation ability to receptors. At Creative Biolabs, you can attain the desirable outcomes with the support of our full-range customized services in a rapid period.
Fig.2 Advantages of our Magic™ in vitro cell-based GPCR functional assay services
Our Magic™ in vitro cell-based GPCR functional assay services can target diverse subtypes and develop experiment designs that hone down on specific receptors. In our Magic™ in vitro cell-based GPCR functional assay services, we target 29 GPCRs and their different subtypes. Here, we provide some targets for your convenience.
Q1: What makes GPCRs such a desirable therapeutic target?
A1: The human genome contains 850 G protein-coupled receptors (GPCRs), with around half of them being potential targets for drug development. Notably, around forty percent of presently available medications interact with GPCRs. This is because GPCRs play a crucial role in regulating various processes in human physiology, such as growth, metabolism, and homeostasis. Due to this, drug development has given great importance to the research and targeting of GPCRs.
At Creative Biolabs, we are always working on improving both our services and our technology in order to remain one step ahead of the competition and to propel forward the process of drug discovery. We continually focus on delivering high-quality outcomes to each of our customers.
If you want to know more details about our Magic™ in vitro cell-based GPCR functional assay services, please don't hesitate to contact us. We sincerely anticipate partnering with you.
Reference
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